Affinity DataKi: 0.380nMAssay Description:Displacement of [3H]raclopride from dopamine D2 receptor in rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.430nMAssay Description:Displacement of [3H]raclopride from dopamine D2 receptor in rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.12nMAssay Description:Displacement of [3H]raclopride from dopamine D2 receptor in rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Displacement of [3H]raclopride from human cloned dopamine D2 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:Displacement of [3H]spiperone from rat dopamine D2 receptor in brain striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 4.10nMAssay Description:Displacement of [3H]spiperone from rat dopamine D2 receptor in brain striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 7.70nMAssay Description:Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 11.1nMAssay Description:Displacement of [3H]raclopride from dopamine D2 receptor in rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [3H]spiperone from rat dopamine D2 receptor in brain striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 17.7nMAssay Description:Displacement of [3H]raclopride from dopamine D2 receptor in rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 19.9nMAssay Description:Displacement of [3H]raclopride from dopamine D2 receptor in rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Displacement of [3H]spiperone from rat dopamine D2 receptor in brain striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cellsMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
University of Debrecen
Curated by ChEMBL
University of Debrecen
Curated by ChEMBL
Affinity DataKi: 31nMAssay Description:Competitive inhibition of rabbit muscle glycogen phosphorylase-b using alpha-D-glucose-1-phosphate as substrate by Dixon plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Displacement of [3H]raclopride from human cloned dopamine D2 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Displacement of [3H]raclopride from rat dopamine D2(short) receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Competitive inhibition of N-terminal His-tagged human OGA using 4-Mu-GlcNAc as substrate assessed as inhibition constant by measuring liberation of n...More data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:Displacement of [3H]raclopride from rat dopamine D2(short) receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 47nMAssay Description:Competitive inhibition of cow HexA/HexB (unknown origin) using pNP-GlcNAc as substrate assessed as inhibition constant by measuring liberation of nit...More data for this Ligand-Target Pair
Affinity DataKi: 48nMAssay Description:Displacement of [3H]spiperone from rat dopamine D2 receptor in brain striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Inhibition of OGA (unknown origin) using pNP-O-GlcNAc as substrate assessed as inhibition constant incubated for 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 54.7nMAssay Description:Displacement of [3H]raclopride from dopamine D2 receptor in rat striatal membraneMore data for this Ligand-Target Pair
Affinity DataKi: 60nMAssay Description:Displacement of [3H]raclopride from rat dopamine D2(short) receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 75nMAssay Description:Displacement of [3H]raclopride from rat dopamine D2(short) receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 78nMAssay Description:Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 78nMAssay Description:Displacement of [3H]spiperone from rat recombinant dopamine D3 receptor expressed in SF9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 83nMAssay Description:Competitive inhibition of N-terminal His-tagged human OGA using 4-Mu-GlcNAc as substrate assessed as inhibition constant by measuring liberation of n...More data for this Ligand-Target Pair
Affinity DataKi: 88nMAssay Description:Displacement of [3H]raclopride from human cloned dopamine D2 receptor expressed in CHO cell membraneMore data for this Ligand-Target Pair
Affinity DataKi: 101nMAssay Description:Displacement of [3H]SCH23390 from dopamine D1 receptor in mouse Ltk- fibroblast cellsMore data for this Ligand-Target Pair
Affinity DataKi: 125nMAssay Description:Competitive inhibition of cow HexA/HexB (unknown origin) using pNP-GlcNAc as substrate assessed as inhibition constant by measuring liberation of nit...More data for this Ligand-Target Pair
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
University of Debrecen
Curated by ChEMBL
University of Debrecen
Curated by ChEMBL
Affinity DataKi: 125nMAssay Description:Competitive inhibition of rabbit muscle glycogen phosphorylase-a in presence of varying levels of glucose-1-phosphate and constant concentration of g...More data for this Ligand-Target Pair
Affinity DataKi: 130nMAssay Description:Inhibition of HexA/HexB (unknown origin)More data for this Ligand-Target Pair
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University of Debrecen
Curated by ChEMBL
University of Debrecen
Curated by ChEMBL
Affinity DataKi: 143nMAssay Description:Competitive inhibition of 6xHis-tagged human liver glycogen phosphorylase-a expressed in Escherichia coli BL21 Gold (DE3) assessed as release of inor...More data for this Ligand-Target Pair
Affinity DataKi: 154nMAssay Description:Competitive inhibition of cow HexA/HexB (unknown origin) using pNP-GlcNAc as substrate assessed as inhibition constant by measuring liberation of nit...More data for this Ligand-Target Pair
Affinity DataKi: 155nMAssay Description:Competitive inhibition of N-terminal His-tagged human OGA using pNP-GlcNAc as chromogenic substrate assessed as inhibition constant by measuring libe...More data for this Ligand-Target Pair
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
University of Debrecen
Curated by ChEMBL
University of Debrecen
Curated by ChEMBL
Affinity DataKi: 160nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase bMore data for this Ligand-Target Pair
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
University of Debrecen
Curated by ChEMBL
University of Debrecen
Curated by ChEMBL
Affinity DataKi: 160nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase b by Dixon plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 167nMAssay Description:Competitive inhibition of N-terminal His-tagged human OGA using pNP-GlcNAc as chromogenic substrate assessed as inhibition constant by measuring libe...More data for this Ligand-Target Pair
Affinity DataKi: 170nMAssay Description:Competitive inhibition of cow HexA/HexB (unknown origin) using pNP-GlcNAc as substrate assessed as inhibition constant by measuring liberation of nit...More data for this Ligand-Target Pair
TargetGlycogen phosphorylase, liver form(Homo sapiens (Human))
University of Debrecen
Curated by ChEMBL
University of Debrecen
Curated by ChEMBL
Affinity DataKi: 172nMAssay Description:Competitive inhibition of human liver glycogen phosphorylase-a assessed as release of inorganic phosphate using varying levels of glucose-1-phosphate...More data for this Ligand-Target Pair
Affinity DataKi: 190nMAssay Description:Competitive inhibition of N-terminal His-tagged human OGA using pNP-GlcNAc as chromogenic substrate assessed as inhibition constant by measuring libe...More data for this Ligand-Target Pair
TargetGlycogen phosphorylase, muscle form(Oryctolagus cuniculus (rabbit))
University of Debrecen
Curated by ChEMBL
University of Debrecen
Curated by ChEMBL
Affinity DataKi: 191nMAssay Description:Competitive inhibition of rabbit muscle glycogen phosphorylase-b in presence of varying levels of glucose-1-phosphate and constant concentration of g...More data for this Ligand-Target Pair
Affinity DataKi: 205nMAssay Description:Competitive inhibition of cow HexA/HexB (unknown origin) using pNP-GlcNAc as substrate assessed as inhibition constant by measuring liberation of nit...More data for this Ligand-Target Pair
Affinity DataKi: 242nMAssay Description:Displacement of [3H]spiperone from rat dopamine D2 receptor in brain striatal membraneMore data for this Ligand-Target Pair